UniProt/SwissProt ID: | MC4R_HUMAN |
Description: | melanocortin 4 receptor [Source:HGNC Symbol;Acc:6932] |
Location: | chr18 q21.32 |
Node attribute: | GPCR; receptor; substrate |
Phosphorylation site |
Position | PhosphoPeptide | Catalytic kinase | Source |
---|---|---|---|
S330 | LCDLSs | ADRBK1 | HPRD |
S329 | GLCDLsS | GRK-2 | phosphoELM |
S330 | LCDLSsRY | PKA_group | RegPhos |
T312 | QELRKtFKEII | GRK_group | phosphoELM; RegPhos |
T312 | QELRKtFKEII | BARK1 | RegPhos |
S330 | LCDLSsRY | BARK1(GRK2 | RegPhos |
Y41 | SDGGCyEQLFV | PhosphoSitePlus | |
T312 | QELRKtFKEII | PhosphoSitePlus | |
S330 | LCDLSsRY | PKACa | RegPhos |
S330 | LCDLSs | GRK_group | phosphoELM |
S329 | GLCDLsS | PRKACA | HPRD |
T312 | QELRKtFKEII | PKA_group | phosphoELM; RegPhos |
S330 | LCDLSsRY | GRK_group | RegPhos |
T312 | QELRKtFKEII | PKACa | RegPhos |
T312 | QELRKtFKEII | ADRBK1 | HPRD |
S329 | GLCDLsS | ADRBK1 | HPRD |
S330 | LCDLSsRY | BARK1 | RegPhos |
S329 | GLCDLsSRY | BARK1(GRK2 | RegPhos |
S329 | GLCDLsSRY__ | PhosphoSitePlus | |
S47 | EQLFVsPEVFV | TM | PhosphoSitePlus |
S330 | LCDLSs | GRK-2 | phosphoELM |
S329 | GLCDLsSRY | GRK_group | RegPhos |
S36 | LGKGYsDGGCY | PhosphoSitePlus | |
S330 | LCDLSs | PRKACA | HPRD |
S330 | LCDLSsRY___ | PhosphoSitePlus | |
S329 | GLCDLsSRY | PKACa | RegPhos |
S330 | LCDLSs | PKA_group | phosphoELM |
S329 | GLCDLsSRY | PKA_group | RegPhos |
T312 | QELRKtFKEII | PRKACA | HPRD |
S329 | GLCDLsSRY | BARK1 | RegPhos |
Y148 | IAVDRyFTIFY | 7tm_1 | PhosphoSitePlus |
S329 | GLCDLsS | PKA_group | phosphoELM |
Y157 | FYALQyHNIMT | 7tm_1 | PhosphoSitePlus |
S329 | GLCDLsS | GRK_group | phosphoELM |
Y35 | SLGKGySDGGC | PhosphoSitePlus | |
Dephosphorylation site |
MC4R_HUMAN do not have dephosphorylation site. |
Mutation site |
Ensembl ID | Variation | Source | Cancer name | Pubmed |
---|---|---|---|---|
ENSP00000299766 | N3K | COSMIC | Ovarian Cancer | 21720365 |
ENSP00000299766 | M161I | COSMIC | Head and Neck Cancer | 21798893 |
ENSP00000299766 | G34R | COSMIC | Lung Cancer | 20668451 |
Differential expressed protein |
MC4R_HUMAN is not differential expressed protein. |
Hyperphosphorylation site |
MC4R_HUMAN do not have hyperphosphorylation site. |
Direct Interaction Pair |
Source | Target | Relationship | Resource |
---|---|---|---|
AGRP_HUMAN | MC4R_HUMAN | ligand -> receptor | HPMR |
MC4R_HUMAN | GNAS1_HUMAN | GPCR -> Gprotein | gpDB |
MC4R_HUMAN | GNAS2_HUMAN | GPCR -> Gprotein | gpDB |
ARBK1_HUMAN | MC4R_HUMAN | kinase -> substrate | RegPhos; Robert H Newman (2013) |
KPCA_HUMAN | MC4R_HUMAN | kinase -> substrate | HPRD |
Function Annotation |
KEGG Pathway |
KEGG ID | Pathway |
---|---|
hsa04080 | Neuroactive ligand-receptor interaction |
Gene Ontology |
GO ID | GO_Term | Evidence | Ontology |
---|---|---|---|
GO:2000252 | negative regulation of feeding behavior | IEA | biological_process |
GO:0045780 | positive regulation of bone resorption | IEA | biological_process |
GO:0031625 | ubiquitin protein ligase binding | IPI | molecular_function |
GO:0006112 | energy reserve metabolic process | IEA | biological_process |
GO:0004930 | G-protein coupled receptor activity | IEA | molecular_function |
GO:0004980 | melanocyte-stimulating hormone receptor activity | IEA | molecular_function |
GO:0016021 | integral to membrane | IEA | cellular_component |
GO:0007186 | G-protein coupled receptor signaling pathway | IEA | biological_process |
GO:0007631 | feeding behavior | IEA | biological_process |
GO:0007188 | adenylate cyclase-modulating G-protein coupled rec | TAS | biological_process |
GO:0019222 | regulation of metabolic process | IEA | biological_process |
GO:0004977 | melanocortin receptor activity | IEA | molecular_function |
GO:0017046 | peptide hormone binding | IEA | molecular_function |
GO:0005634 | nucleus | IEA | cellular_component |
GO:0005515 | protein binding | IPI | molecular_function |
GO:0032868 | response to insulin stimulus | IEA | biological_process |
GO:0004980 | melanocyte-stimulating hormone receptor activity | IPI | molecular_function |
GO:0002024 | diet induced thermogenesis | IEA | biological_process |
GO:0004977 | melanocortin receptor activity | TAS | molecular_function |
GO:0030819 | positive regulation of cAMP biosynthetic process | IDA | biological_process |
GO:0005515 | protein binding | IEA | molecular_function |
GO:0005886 | plasma membrane | TAS | cellular_component |
GO:0042923 | neuropeptide binding | IPI | molecular_function |
GO:0030073 | insulin secretion | IEA | biological_process |
GO:0045780 | positive regulation of bone resorption | IMP | biological_process |